| New deuterated trihexyphenidyl compound is prepared by refluxing piperidine salt with benzaldehyde compound and ketone compound in presence of acid, reacting obtained substituted piperidinyl compound with halobenzene compound in presence of metal catalyst and initiator | |
| 2024-01-25 | |
| 专利权人 | CLEARSYNTH LABS LTD (CLEA-Non-standard) |
| 申请日期 | 2024-01-25 |
| 专利号 | IN202421005224-A |
| 成果简介 | NOVELTY - Deuterated trihexyphenidyl compound (I), or its salt is new. USE - Deuterated trihexyphenidyl compound. ADVANTAGE - The compound (I) ensures improved efficacy, reduced side effects, improved bioavailability, prolonged duration of action, and less susceptible to certain types of drug interactions, and can be prepared with yield of 50-99%, and purity of 80-99%. DETAILED DESCRIPTION - Deuterated trihexyphenidyl compound of formula (I), or its salt is new. R1-R22=H, D, 1-5C alkyl, or aryl. An INDEPENDENT CLAIM is included for a method for preparing (I). |
| IPC 分类号 | C07D-207/04 ; C07D-207/08 |
| 国家 | 印度 |
| 专业领域 | 医药卫生 |
| 语种 | 英语 |
| 成果类型 | 专利 |
| 文献类型 | 科技成果 |
| 条目标识符 | http://119.78.100.226:8889/handle/3KE4DYBR/18339 |
| 专题 | 中国科学院新疆生态与地理研究所 |
| 作者单位 | CLEARSYNTH LABS LTD (CLEA-Non-standard) |
| 推荐引用方式 GB/T 7714 | MODALA R,JONNALAGADDA R N S,SAKTHIVEL K,et al. New deuterated trihexyphenidyl compound is prepared by refluxing piperidine salt with benzaldehyde compound and ketone compound in presence of acid, reacting obtained substituted piperidinyl compound with halobenzene compound in presence of metal catalyst and initiator. IN202421005224-A[P]. 2024. |
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