| 4-((ARYL)(METHYL)AMINO)QUINAZOLINE-7-CARBOXYLIC ACID DERIVATIVES WITH ANTI-TUMOUR ACTION AND METHOD FOR PRODUCTION THEREOF | |
| 2024-07-10 | |
| 专利权人 | FEDERAL STATE BUDGETARY INST (FSBI-C) |
| 申请日期 | 2024-07-10 |
| 专利号 | RU2834688-C1 |
| 成果简介 | NOVELTY - Invention relates to 4-((aryl)(methyl)amino)quinazoline-7-carboxylic acid derivatives having the following general formula: , where R1 is hydrogen or methyl, R2 is hydrogen or OMe, A is -(CH2)5- or para-phenylene (-C4H6-), as well as methods of their production. USE - Chemistry. ADVANTAGE - Novel compounds are obtained, which have inhibitory activity on histone deacetylase (HDAC) and can be used in medicine for treating oncological diseases. 3 cl, 1 tbl, 1 dwg, 20 ex |
| IPC 分类号 | A61K-031/517 ; A61P-035/00 ; C07D-239/94 |
| 国家 | 俄罗斯 |
| 专业领域 | 化学化工 |
| 语种 | 英语 |
| 成果类型 | 专利 |
| 文献类型 | 科技成果 |
| 条目标识符 | http://119.78.100.226:8889/handle/3KE4DYBR/15867 |
| 专题 | 中国科学院新疆生态与地理研究所 |
| 作者单位 | FEDERAL STATE BUDGETARY INST (FSBI-C) |
| 推荐引用方式 GB/T 7714 | BORISOVA L M,OSIPOV V N,GUSEV D V,et al. 4-((ARYL)(METHYL)AMINO)QUINAZOLINE-7-CARBOXYLIC ACID DERIVATIVES WITH ANTI-TUMOUR ACTION AND METHOD FOR PRODUCTION THEREOF. RU2834688-C1[P]. 2024. |
| 条目包含的文件 | 条目无相关文件。 | |||||
除非特别说明,本系统中所有内容都受版权保护,并保留所有权利。
修改评论